Thursday September 17, 2015 |
08:15 | Coffee - Registration |
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08:50 | Welcome and Opening |
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| Keynote Lecture |
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08:55 | We Urgently Need More Medicinal Chemists to Generate Novel Tools to Dissect Disease Biology, and New Drugs for Patients |
Prof. Chas BOUNTRA (UNIVERSITY OF OXFORD, Oxford, United Kingdom) |
| EFMC-YMCS Competition Presentation Session I |
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09:40 | Innovative Oligourea Foldamers with Antimicrobial Effects : Application to Bacillus Anthracis Infection
Winner of the young medicinal chemist meeting in France |
Ms Stéphanie ANTUNES (UNIVERSITÉ DE BORDEAUX, Pessac, France) |
10:00 | Novel SAM Analogues for Sequence-Specific DNA Labeling
Winner of the young medicinal chemist meeting in Belgium (KVCV) |
Ms Charlotte VRANKEN (KULEUVEN, Heverlee, Belgium) |
10:20 | Finding Novel Treatments Against Neglected Parasitic Diseases Using Target Repurposing of Phosphodiesterases |
Dr Ewald EDINK (VU UNIVERSITY AMSTERDAM, Delft, The Netherlands) |
10:40 | Coffee Break |
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| EFMC-YMCS Competition Presentation Session II |
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11:05 | Synthesis of Novel Pyrido[1,2-c]Pyrimidine Derivatives - 5-HT1A Receptors
and Serotonin Transporter Ligands
Winner of the young medicinal chemist meeting in Poland |
Ms Anna GOMOLKA (MEDICAL UNIVERSITY OF WARSAW, Warsaw, Poland) |
11:25 | Development of Pharmacological Tools to Explore the Orphan G Protein-coupled Receptor GPR35
Winner of the young medicinal chemist meeting in Germany |
Dr Dominik THIMM (UNIVERSITÄT BONN, Bonn, Germany) |
11:45 | Binding Kinetics at the GnRH Receptor - A Comparison of Three Different Assays
Winner of the young medicinal chemist meeting in The Netherlands |
Ms Indira NEDERPELT (UNIVERSITY OF LEIDEN, Leiden, The Netherlands) |
12:05 | Photoisomerizable Phenylazopyridines Enable the Control of Metabotropic Glutamate Receptor Subtpe 5 Activity with Light |
Mr Xavier GÓMEZ-SANTACANA (INSTITUTE FOR ADVANCED CHEMISTRY OF CATALONIA - CSIC, Amsterdam, The Netherlands) |
12:25 | Flash Poster Presentations |
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Dr Filipe ELVAS (UNIVERSITY OF ANTWERP, Wilrijk, Belgium) |
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Dr Bhatia SUMATI  (FREE UNIVERSITY OF BERLIN, Berlin, Germany) |
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Dr Kuntarat ARUNRUNGVICHIAN (MAHIDOL UNIVERSITY, Bangkok, Thailand) |
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Ms Ramatoulie CAMARA (UNIVERSITY OF HERTFORDSHIRE, Hatfield, United Kingdom) |
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Dr Rafaela GLADYSZ (UANTWERP, Antwerpen, Belgium) |
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Mr Marton VASS (VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands) |
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Ms Leticia MONJAS GOMEZ (UNIVERSITY OF GRONINGEN, Groningen, The Netherlands) |
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Dr Andrea PINTO (UNIVERSITY OF MILAN, Milan, Italy) |
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Mr Maciej ROGACKI (UNIVERSITY OF ANTWERP, Antwerp, Belgium) |
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Dr Stefano SAINAS (UNIVERSITY OF TORINO, Torino, Italy) |
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Prof. Dmitry TSVELIKHOVSKY (THE HEBREW UNIVERSITY OF JERUSALEM, Jerusalem, Israel) |
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Ms Hannah WAPENAAR (RIJKSUNIVERSITEIT GRONINGEN, Groningen, The Netherlands) |
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Dr Thomas STORR (UNIVERSITY OF NOTTINGHAM, Nottingham, United Kingdom) |
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Dr Tina RITSCHEL (CMBI 260 / RADBOUDUMC, Nijmegen, The Netherlands) |
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Ms Anne FRANK (FREIE UNIVERSITÄT BERLIN, Berlin, Germany) |
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Mr Edwin KROON (UNIVERSITY OF GRONINGEN, Groningen, The Netherlands) |
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Mr Girdhar SINGH DEORA (THE UNIVERSITY OF QUEENSLAND, Australia) |
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Dr Irene GARCIA SALADO (UNIVERSITY OF ANTWERP, Antwerpen, Belgium) |
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Ms Leena KEURULAINEN (UNIVERSITY OF HELSINKI, Helsinki, Finland) |
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Ms Natalie THEODOULOU (GLAXOSMITHKLINE, Stevenage, United Kingdom) |
13:05 | EFMC-YMCS Poster Session and Lunch |
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| EFMC-YMCS Competition Presentation Session III |
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15:05 | Cathepsin B Inhibitors Impair the Processes of Tumour Progression
Winner of the young medicinal chemist meeting in Slovenia
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Dr Izidor SOSIC (UNIVERSITY OF LJUBLJANA, Ljubljana, Slovenia) |
15:25 | SWI/SNF Bromodomain Inhibitor Development and Testing in SWI/SNF Mutant Cancers
Winner of the young medicinal chemist meeting in the United Kingdom |
Ms Charlotte SUTHERELL (UNIVERSITY OF CAMBRIDGE, Cambridge, United Kingdom) |
15:45 | Nortopsentin Analogues with Potent Activity against Diffuse Malignant Peritoneal Mesothelioma (DMPM)
Winner of the young medicinal chemist meetings in Italy |
Mrs Barbara PARRINO (UNIVERSITY OF PALERMO (1), PALERMO , Italy) |
16:05 | 2-(4΄-Aminophenyl)Benzothiazole Derivatives As Pharmacophores In Tricarbonyl M(Co)3+ (M = Re, 99mtc) Complexes For Tumor Diagnosis And Therapy
Winner of the young medicinal chemist meeting in Greece |
Mr Alexandros STOURAITIS (NCSR DEMOKRITOS, Athens, Greece) |
16:25 | Coffee Break |
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| EFMC-YMCS Competition Presentation Session IV |
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16:40 | Iminoboronates as a Novel Bioconjugation Method
Winner of the young medicinal chemist meeting in Portugal |
Dr Pedro CAL (UNIVERSITY OF LISBON, Lisboa, Portugal) |
17:00 | Novel CF3-Containing Pyrrolidones as Amidine-based BACE1 Inhibitors
Winner of the young medicinal chemist meeting in Spain |
Mrs Myriam CIORDIA JIMENEZ (UNIVERSIDAD CEU SAN PABLO, Madrid, Spain) |
17:20 | Playing Properties Right in the CD38 FBDD Programme: Small Changes Produced Significant Shifts in Property profiles |
Mr Ben WHITEHURST (GLAXOSMITHKLINE, Stevenage, United Kingdom) |
17:40 | Networking Break |
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17:55 | Closing and Award Ceremony |
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18:15 | EFMC-YMCS Networking and Drinks |
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